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This book compares empirical discovery methods for biologically relevant molecules with serendipitous discovery and rational design, and highlights the general approach to empirical discovery and its advantanges/disadvantages. It provides a comprehensive and logical look at experimental methods for discovery of biologically relevant molecules, and includes sections on pragmatic molecular discovery, finding useful natural molecules, empirical methods, directed evolution, high-throughput synthesis and screening, rational molecular design, empirical versus rational design, and the limits of empirical methods.